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    Título
    Plasma protein binding of levamisole in several species
    Autor
    Sahagún, Ana M.
    Fernández, Nélida
    Terán, M. TeresaAutoridad Buleria
    García, Juan J.
    Sierra, MatildeAutoridad BuleriaORCID
    Diez, M. José
    Facultad/Centro
    Facultad de Veterinaria
    Área de conocimiento
    Farmacologia
    Datos de la obra
    Methods and Findings in Experimental and Clinical Pharmacology, 1997, vol. 19, n. 3
    Editor
    Prous Science
    Fecha
    1997-02-14
    Abstract
    The binding of levamisole to total plasma proteins of 6 animal species was determined in vitro by equilibrium dialysis. The percentage of bound drug protein was independent of levamisole concentration within the range studied, 5-50µg/ml (ANOVA). Levamisole was bound to a low extent to plasma proteins of each animal species (19.40-25.91%). There were significant differences in the extent of levamisole binding among species (ANOVA). Owing to the low degree of protein binding and the high volume of distribution of levamisole, the variations in protein binding due to different factors would not be of major clinical importance in its therapeutic application.
    Materia
    Ecología. Medio ambiente
    Farmacología
    Veterinaria
    Palabras clave
    Levamisole
    Protein binding
    Equilibrium dialysis
    Peer review
    SI
    URI
    http://hdl.handle.net/10612/4575
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    Methods and Findings in Experimental and Clinical Pharmacology, 1997, p. 185-187
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