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    Título
    Effect of bovine ABCG2 Y581S polymorphism on concentrations in milk of enrofloxacin and its active metabolite ciprofloxacin
    Autor
    Merino Peláez, GraciaAutoridad BuleriaORCID
    Álvarez de Felipe, Ana IsabelAutoridad BuleriaORCID
    Prieto Fernández, Julio GabrielAutoridad BuleriaORCID
    Fuente, Álvaro de la
    García Mateos, Dafne
    Otero, Jon Andoni
    Facultad/Centro
    Facultad de Veterinaria
    Área de conocimiento
    Fisiologia
    Datos de la obra
    Journal of Dairy Science, 2016, vol. 99, n. 7
    Editor
    Elsevier
    Fecha
    2016
    Abstract
    The ATP-binding cassette transporter G2 (ABCG2) is involved in the secretion of several drugs into milk. The bovine Y581S ABCG2 polymorphism increases the secretion into milk of the fluoroquinolone danofloxacin in Holstein cows. Danofloxacin and enrofloxacin are the fluoroquinolones most widely used in veterinary medicine. Both enrofloxacin (ENRO) and its active metabolite ciprofloxacin (CIPRO) reach milk at relatively high concentrations. The aim of this work was to study the effect of the bovine Y581S ABCG2 polymorphism on in vitro transport as well as on concentrations in plasma and in milk of ENRO and CIPRO. Experiments using cells over-expressing bovine ABCG2 showed the effects of ABCG2 on the transport of CIPRO demonstrating more efficient in vitro transport of this antimicrobial by the S581 variant
    Materia
    Veterinaria
    Palabras clave
    Bovine ABCG2
    Polymorphism
    Enrofloxacin
    Ciprofloxacin
    Peer review
    SI
    URI
    http://hdl.handle.net/10612/6862
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